SCHEMBL10522151

SCHEMBL10522151

Cc1[nH]cnc1CC1CC(OC(=O)/C=C\C(=O)OC2CC(Cc3nc[nH]c3C)C(=O)c3c2n(C)c2ccccc32)c2c(c3ccccc3n2C)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.44
CYP3A4 P08684 3/20 0.44
KCNH2 Q12809 3/20 0.44
CYP1A2 P05177 2/20 0.44
HTR2B P41595 2/20 0.44
ADRA2C P18825 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1A P35348 1/20 0.44
CASP6 P55212 1/20 0.43
HTR3E A5X5Y0 3/20 0.40
HTR3B O95264 3/20 0.40
HTR3D Q70Z44 3/20 0.40
HTR3C Q8WXA8 3/20 0.40
NPY1R P25929 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
SLC22A3 O75751 1/20 0.35
CHRNB2 P17787 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9597521 0.90 HTR3A (0.34) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597379 0.89 HTR3A (0.33) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9596742 0.88 HTR3A (0.38) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597424 0.88 HTR3A (0.33) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597678 0.88 HTR3A (0.38) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9596524 0.88 HTR3A (0.36) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597348 0.88 HTR3A (0.36) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597198 0.87 HTR3A (0.35) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9596051 0.87 P2RX7 (0.34) HTR3ACYP3A4KCNH2CYP1A2HTR2B
SCHEMBL9597016 0.86 HTR6 (0.36) HTR3ACYP3A4KCNH2CYP1A2HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4859662-A Tetrahydro-imidazolylmethylcarbazolones and analogs thereof for treating 5-HT function disturbances GLAXO GROUP LIMITED (GB) 1989-08-22 US disclosed
US-4822881-A PSYCHOTIC DISORDERS, ANXIETY, NAUSEA, VOMITING GLAXO GROUP LIMITED 1989-04-18 US disclosed