SCHEMBL10522299

SCHEMBL10522299

CC(C)(C)OC(=O)c1nnnn1CN

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
MAPK1 P28482 1/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 2/20 0.32
GAA P10253 2/20 0.32
HPGD P15428 2/20 0.32
HIF1A Q16665 2/20 0.32
THRB P10828 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
GHSR Q92847 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10840248 0.65 MAPK1 (0.44) FAAHMAPK1MAPTKDM4EALDH1A1
SCHEMBL6581440 0.63 FAAH (0.58) FAAHMAPTSMN1; SMN2
SCHEMBL11332477 0.63 FAAH (0.37) FAAHMAPK1GHSRKMT2A
SCHEMBL18839755 0.62 MAPK1 (0.44) MAPK1MAPTKDM4EALDH1A1GAA
SCHEMBL10128478 0.62 MAPK1 (0.41) FAAHMAPK1MAPTKDM4EALDH1A1
SCHEMBL11778347 0.61 MAPK1 (0.69) MAPK1MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL11776322 0.61 MAPK1 (0.51) MAPK1MAPTALDH1A1GAAHPGD
SCHEMBL20128067 0.61 MAPK1 (0.33) FAAHMAPK1ALDH1A1HPGDSMN1; SMN2
SCHEMBL20518647 0.61 CA1 (0.38) FAAHMAPK1MAPTALDH1A1GLA
SCHEMBL18839913 0.61 MAPK1 (0.47) MAPK1MAPTKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4829053-A Amino acid derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-05-09 US disclosed
EP-0262318-A2 Renin-inhibiting amino acid derivatives MERCK PATENT GmbH (DE) 1988-04-06 EP disclosed