SCHEMBL10528166

SCHEMBL10528166

O=c1ccc2cnc3ncccc3c2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.41
PARP1 P09874 4/20 0.38
LMNA P02545 1/20 0.38
CA12 O43570 4/20 0.38
CA9 Q16790 4/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
AURKA O14965 1/20 0.37
FGFR1 P11362 1/20 0.35
FLT1 P17948 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CA1 P00915 1/20 0.34
CA3 P07451 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29611187 0.77 KDM4E (0.48) PARP1CA12CA9KDM4ECA1
SCHEMBL22607244 0.77 KDM4E (0.48) PARP1CA12CA9KDM4ECA1
SCHEMBL4464552 0.77 MAPT (0.50) PARP1LMNACA12CA9AURKA
SCHEMBL8600442 0.76 AXL (0.46) HCAR2PARP1LMNAKDM4EMAPT
SCHEMBL28115036 0.73 CA12 (0.41) CA12CA9KDM4EMEN1ALDH1A1
SCHEMBL730906 0.73 LMNA (0.42) HCAR2PARP1LMNAAURKAFGFR1
SCHEMBL30846772 0.72 PARP1 (0.42) HCAR2PARP1LMNACA12CA9
SCHEMBL1982985 0.71 CYP3A4 (0.47) PARP1LMNAAURKAKDM4EMEN1
SCHEMBL13629310 0.69 ALDH1A1 (0.43) HCAR2PARP1LMNAAURKAKDM4E
SCHEMBL29871779 0.69 MAPT (0.54) LMNACA12CA9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4801590-A ANGINA, ANTICANCER, CARDIOVASCULAR DISORDERS, HEADACHES, PSORIASIS, ASTHMA, ANTICOAGULANTS BEIERSDORF AG (DE) 1989-01-31 US disclosed
EP-0253171-A1 Pyrido[1,8]naphthyridinones, process for their preparation and their use and compositions containing them Beiersdorf-Lilly GmbH (DE) 1988-01-20 EP disclosed