SCHEMBL10529985

SCHEMBL10529985

C=C(C(=O)c1ccc(Cl)cc1Cl)n1cncn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.61
ALDH1A1 P00352 5/20 0.56
MAPT P10636 4/20 0.56
LMNA P02545 4/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
HTT P42858 1/20 0.56
TSHR P16473 3/20 0.49
HPGD P15428 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
GABRA1 P14867 1/20 0.49
GABRG2 P18507 1/20 0.49
GABRB3 P28472 1/20 0.49
PKM P14618 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
HSP90AA1 P07900 1/20 0.45
MAPK1 P28482 1/20 0.45
USP2 O75604 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080873 0.77 ALDH1A1 (0.73) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11087065 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL10946350 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11150916 0.77 ALDH1A1 (0.73) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL10946345 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11087066 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11228351 0.74 ALDH1A1 (0.51) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11228340 0.74 ALDH1A1 (0.51) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL11432191 0.74 ALDH1A1 (0.51) CYP19A1ALDH1A1MAPTLMNAMEN1
SCHEMBL10528860 0.74 CYP19A1 (0.48) CYP19A1ALDH1A1MAPTLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183494-B1 TRIAZOLE ANTIFUNGAL AGENTS Pfizer Limited (GB) 1989-01-11 EP disclosed
US-4767777-A Triazole antifungal agents PFIZER INC. (US) 1988-08-30 US disclosed
EP-0164246-B1 TRIAZOLE ANTIFUNGAL AGENTS Pfizer Limited (GB) 1988-08-10 EP disclosed
US-4618616-A MAMMALS AND PLANTS; 1,2,4-TRIAZOLE DI-SUBSTITUTED PFIZER INC. (US) 1986-10-21 US disclosed
EP-0183494-A2 Triazole antifungal agents Pfizer Limited (GB) 1986-06-04 EP disclosed
EP-0164246-A2 Triazole antifungal agents Pfizer Limited (GB) 1985-12-11 EP disclosed