SCHEMBL10544477

SCHEMBL10544477

CCOc1ncccc1C1OC(=O)NC1=O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.42
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 4/20 0.35
P2RX3 P56373 3/20 0.35
TSHR P16473 3/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
NPC1 O15118 2/20 0.34
PPARG P37231 2/20 0.34
HPGD P15428 2/20 0.34
RAB9A P51151 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10544451 0.86 CA2 (0.50) CA2P2RX3
SCHEMBL11040310 0.79 CA2 (0.51) CA2ALDH1A1TSHRGAAHTT
SCHEMBL10546481 0.76 CA2 (0.40) CA2L3MBTL1PPARGPPARDPPARA
SCHEMBL10547400 0.76 CA2 (0.40) CA2PPARGPPARDPPARA
SCHEMBL10547592 0.73 CA2 (0.45) CA2ALDH1A1TSHRGAAHTT
SCHEMBL28861148 0.70 PDE1A (0.37) ALDH1A1L3MBTL1P2RX3TSHRNPC1
SCHEMBL10892219 0.69 CA2 (0.44) CA2ALDH1A1GAAPPARGPPARD
SCHEMBL11040283 0.69 CA2 (0.47) CA2ALDH1A1L3MBTL1TSHRPPARG
SCHEMBL11040416 0.69 HTR2C (0.48) CA2TSHRGAAPPARGHPGD
SCHEMBL11038153 0.69 CA2 (0.43) CA2L3MBTL1PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4812471-A Hypoglycemic 5-(isoxazolyl or isothiazolyl)-oxazolidine-2,4-diones PFIZER INC. (US) 1989-03-14 US disclosed
US-4753956-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1988-06-28 US disclosed
US-4689336-A Hypoglycemic 5-substituted oxazolidine 2,4-diones PFIZER INC. (US) 1987-08-25 US disclosed
US-4565820-A ANTIDIABETIC AGENTS PFIZER INC. (US) 1986-01-21 US disclosed
US-4431810-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1984-02-14 US disclosed
US-4342771-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1982-08-03 US disclosed