SCHEMBL10548754

SCHEMBL10548754

CC(CC(=O)O)C(=O)c1ccc(OCCCBr)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
RARB P10826 1/20 0.45
GAA P10253 1/20 0.44
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
PLA2G4B P0C869 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PPARA Q07869 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP13 P45452 1/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733588 0.86 MAPT (0.45) MAPK1L3MBTL1POLBRARBGAA
SCHEMBL10555616 0.84 MAPT (0.49) MAPK1L3MBTL1POLBTDP1RARB
SCHEMBL10557960 0.82 ALDH1A1 (0.54) MAPK1TSHRPLA2G4BALDH1A1MAPT
SCHEMBL10353455 0.79 HDAC3 (0.49) L3MBTL1ALDH1A1MMP9MAPT
SCHEMBL10456769 0.79 ALDH1A1 (0.40) ALDH1A1MMP9
SCHEMBL8213432 0.79 ALDH1A1 (0.54) POLBTDP1ALDH1A1MAPTHTT
SCHEMBL10561154 0.78 CYP19A1 (0.46) MAPK1POLBTDP1GAATSHR
SCHEMBL8787577 0.78 L3MBTL1 (0.49) MAPK1L3MBTL1RARBGAATP53
SCHEMBL6803381 0.77 MAOB (0.61) L3MBTL1PLA2G4BALDH1A1HTT
SCHEMBL9733516 0.77 L3MBTL1 (0.47) MAPK1L3MBTL1RARBGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4857659-A Stereoselective synthesis of leukotriene antagonists MERCK FROSST CANADA, INC. (CA) 1989-08-15 US disclosed
EP-0244164-A1 Stereoselective synthesis of leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1987-11-04 EP disclosed
EP-0236618-A2 Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-09-16 EP disclosed