SCHEMBL10550076

SCHEMBL10550076

O=C(CCS)NC1(C(=O)O)CCCC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
CTSB P07858 2/20 0.36
CTSS P25774 1/20 0.36
CTSL P07711 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MME P08473 2/20 0.33
SHMT1 P34896 2/20 0.33
SHMT2 P34897 2/20 0.33
CYP1A2 P05177 1/20 0.32
FABP4 P15090 3/20 0.31
FABP5 Q01469 3/20 0.31
CYP2C19 P33261 1/20 0.31
SPHK1 Q9NYA1 1/20 0.31
ACE P12821 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10594469 0.79 CTSB (0.38) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL500447 0.78 SPHK1 (0.49) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL13502694 0.77 CTSB (0.36) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL9671904 0.77 SPHK1 (0.48) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL4764313 0.77 CNR2 (0.42) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL8485391 0.76 CNR2 (0.39) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL8683974 0.74 CYP2C19 (0.36) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL14088075 0.74 CYP1A2 (0.38) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL7439122 0.74 CTSB (0.46) CYP4F2CYP4A11CTSBCTSSCTSL
SCHEMBL4317114 0.74 CTSL (0.63) CTSBCTSLALDH1A1SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833152-A Anti-hypertensive agents UNIVERSITY OF MIAMI (US) 1989-05-23 US disclosed
US-4745124-A THIO/ESTER PEPTIDES UNIVERSITY OF MIAMI (US) 1988-05-17 US disclosed
US-4734420-A INHIBITORS OF ANGIOTENSIN CONVERTING ENZYME UNIVERSITY OF MIAMI (US) 1988-03-29 US disclosed
US-4692458-A Anti-hypertensive agents UNIVERSITY OF MIAMI (US) 1987-09-08 US disclosed
US-4690936-A AMINO ACIDS, THIOESTER LINKAGE; ANGIOTENSIN INHIBITORS UNIVERSITY OF MIAMI (US) 1987-09-01 US disclosed
EP-0036713-B1 ANGIOTENSIN CONVERTING ENZYME INHIBITORS UNIVERSITY OF MIAMI (US) 1984-01-18 EP disclosed
EP-0036713-A2 Angiotensin converting enzyme inhibitors UNIVERSITY OF MIAMI (US) 1981-09-30 EP disclosed
US-4108886-A Thiopropanoylamino acid derivatives E. R. SQUIBB & SONS, INC. (US) 1978-08-22 US disclosed