SCHEMBL10552149

SCHEMBL10552149

O=C(O)c1cccc2cc(-c3ccc(Cl)cc3)oc12

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ERAP1 Q9NZ08 12/20 0.66
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
CYSLTR1 Q9Y271 1/20 0.48
CYP1A1 P04798 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP1B1 Q16678 1/20 0.47
AR P10275 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8155546 0.88 MAOA (0.58) ERAP1NPC1RAB9ACYSLTR1
SCHEMBL10546844 0.85 ERAP1 (0.53) ERAP1NPC1RAB9ACYSLTR1AR
SCHEMBL10989066 0.82 CYSLTR1 (0.71) ERAP1NPC1RAB9ACYSLTR1CYP1A1
SCHEMBL10549952 0.82 L3MBTL1 (0.52) ERAP1NPC1RAB9ACYSLTR1CYP1A2
SCHEMBL10551657 0.82 NTRK1 (0.57) ERAP1NPC1RAB9ACYSLTR1CYP1A1
SCHEMBL10547237 0.81 MAOA (0.56) ERAP1NPC1CYSLTR1AR
Hydrochloric Acid SCHEMBL10991396 0.81 CYSLTR1 (0.70) ERAP1NPC1RAB9ACYSLTR1CYP1A1
SCHEMBL5123750 0.78 MCL1 (0.52) ERAP1NPC1RAB9ACYSLTR1
SCHEMBL27974835 0.78 MAOA (0.50) ERAP1
SCHEMBL10549752 0.78 PTGER1 (0.55) ERAP1NPC1RAB9ACYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4882340-A INHIBITS REFLECTIVE CONTRACTION OF URINARY BLADDER TANABE SEIYAKU CO., LTD. (JP) 1989-11-21 US disclosed
US-4829067-A INHIBITORS OF REFLECTIVE CONTRACTION OF BLADDER TANABE SEIYAKU CO., LTD. (JP) 1989-05-09 US disclosed
EP-0306226-A2 A benzofuran derivative and processes for preparing the same Tanabe Seiyaku Co., Ltd. (JP) 1989-03-08 EP disclosed
EP-0270342-A2 A benzo-furan (or -thiophene) derivative and processes for preparing the same Tanabe Seiyaku Co., Ltd. (JP) 1988-06-08 EP disclosed