SCHEMBL10552437

SCHEMBL10552437

COc1ccc(N2C(=O)c3ccccc3C2(C)CC(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.55
NPC1 O15118 8/20 0.51
RAB9A P51151 8/20 0.51
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
GAA P10253 1/20 0.51
RECQL P46063 1/20 0.51
HPGD P15428 2/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NR1H3 Q13133 1/20 0.43
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
MAPT P10636 2/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
PLA2G1B P04054 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14663931 0.74 RAB9A (0.52) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL16155526 0.73 PGR (0.51) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL10651704 0.72 ALDH1A1 (0.48) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL10555272 0.71 SMN1; SMN2 (0.42) PGRKDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL11988993 0.71 NPC1 (0.46) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL10556389 0.71 KDM4E (0.43) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL10553937 0.70 PGR (0.44) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL30667104 0.70 RAB9A (0.52) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL29127949 0.70 RAB9A (0.52) PGRNPC1RAB9AKDM4EALDH1A1
SCHEMBL6088862 0.69 KDM4E (0.56) PGRNPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4879293-A NERVOUS SYSTEM AND PSYCHOSOMATIC DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-07 US disclosed
US-4788191-A ANTIANXIETY AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-11-29 US disclosed
US-4590189-A ANTIANXIETY AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-05-20 US disclosed
EP-0091241-A2 Condensed pyrrolinone derivatives, and their production Takeda Chemical Industries, Ltd. (JP) 1983-10-12 EP disclosed