SCHEMBL10554382

SCHEMBL10554382

Nc1nc2cc3oc(=O)[nH]c3cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP6 P51161 2/20 0.47
KMO O15229 1/20 0.47
NOS1 P29475 4/20 0.41
NOS3 P29474 3/20 0.41
NOS2 P35228 3/20 0.41
BLM P54132 2/20 0.41
PLAU P00749 1/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
BACE1 P56817 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
ADRA2A P08913 1/20 0.41
TSHR P16473 1/20 0.41
THPO P40225 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDE3B Q13370 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9678466 0.80 NOS1 (0.49) KMONOS1NOS3NOS2BLM
SCHEMBL9678778 0.80 KMO (0.47) KMONOS1NOS3NOS2BLM
SCHEMBL10556198 0.80 KMO (0.47) KMONOS1NOS3NOS2BLM
SCHEMBL10552171 0.76 HPGD (0.45) KMONOS1NOS3NOS2BLM
SCHEMBL10551103 0.76 GAA (0.51) KMONOS1NOS3NOS2BLM
SCHEMBL9679002 0.76 KDM4E (0.53) KMONOS1NOS3NOS2BLM
SCHEMBL10557333 0.76 LMNA (0.50) KMONOS1NOS3NOS2BLM
SCHEMBL30295627 0.75 KMO (0.68) KMONOS1NOS3NOS2BLM
SCHEMBL10550319 0.75 KMO (0.42) KMONOS1NOS3NOS2BLM
SCHEMBL9679533 0.74 NPC1 (0.49) PLAUTSHRALDH1A1OGTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831032-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE, ISOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1989-05-16 US disclosed
EP-0207483-A2 Benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1987-01-07 EP disclosed