SCHEMBL10560010

SCHEMBL10560010

CS(=O)(=O)N(Cc1cccnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 18/20 0.57
HDAC1 Q13547 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
HDAC5 Q9UQL6 1/20 0.56
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6733966 0.85 GRM2 (0.60) GRM2
SCHEMBL6734090 0.83 GRM2 (0.66) GRM2HDAC1HDAC6HDAC5
SCHEMBL10556546 0.81 GRM2 (0.65) GRM2CYP3A4
SCHEMBL10557732 0.79 GRM2 (0.54) GRM2CYP3A4
SCHEMBL6727812 0.78 GRM2 (0.81) GRM2
SCHEMBL10556648 0.77 CYP3A4 (0.67) GRM2CYP3A4
SCHEMBL10559397 0.77 GRM2 (0.61) GRM2CYP3A4
SCHEMBL10559014 0.76 KMT2A (0.55) GRM2
SCHEMBL10558724 0.76 CYP3A4 (0.56) GRM2CYP3A4
SCHEMBL10561180 0.76 LMNA (0.68) GRM2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4874775-A INHIBIT PHYTOPATHOGENS ELI LILLY AND COMPANY (US) 1989-10-17 US disclosed
EP-0206581-A2 Agriculturally-useful sulfonamides ELI LILLY AND COMPANY (US) 1986-12-30 EP disclosed