SCHEMBL10561978

SCHEMBL10561978

CCCCn1c(=O)cc(Cl)n(Cc2ccc(OC)cc2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 1/20 0.48
ADORA3 P0DMS8 5/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALOX15 P16050 1/20 0.43
CMA1 P23946 1/20 0.43
PDE1A P54750 2/20 0.42
PDE1B Q01064 2/20 0.42
PDE1C Q14123 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
P2RX4 Q99571 1/20 0.42
ADORA1 P30542 1/20 0.42
RGS4 P49798 2/20 0.41
RGS8 P57771 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL325735 0.88 MAPT (0.51) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL23679701 0.87 MAPT (0.47) PROKR1ALDH1A1MAPTKDM4EALOX15
SCHEMBL10558278 0.83 PROKR1 (0.49) PROKR1ADORA3ALDH1A1MAPTKDM4E
SCHEMBL320830 0.83 RGS4 (0.53) ADORA3ALDH1A1MAPTKDM4EALOX15
SCHEMBL4847620 0.82 ALDH1A1 (0.50) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL19073410 0.79 MAPT (0.47) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL19073042 0.79 P2RX3 (0.47) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL10502022 0.77 ADORA2A (0.44) ALDH1A1RGS4RGS8GSK3B
SCHEMBL19147820 0.76 KAT2B (0.47) ALDH1A1ALOX15
SCHEMBL31213513 0.75 HPGD (0.52) ADORA3MAPTMEN1KMT2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4824848-A TREATMENT, PREVENTION OF NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-04-25 US disclosed
EP-0237289-A2 Pyrazolo [3,4-d] pyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-09-16 EP disclosed