SCHEMBL10567296

SCHEMBL10567296

CC1(C)C(=O)Nc2cc3c(cc21)NC(c1cn[nH]c1)N3

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.40
PDE3B Q13370 11/20 0.37
PDE3A Q14432 11/20 0.37
PDE4A P27815 10/20 0.37
PDE4B Q07343 10/20 0.37
PDE4C Q08493 10/20 0.37
PDE4D Q08499 10/20 0.37
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
PGR P06401 4/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
BMPR1B O00238 1/20 0.32
BMPR1A P36894 1/20 0.32
TGFBR1 P36897 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567841 0.81
SCHEMBL10567457 0.80 ADORA2B (0.33)
SCHEMBL10566666 0.80 ATAD2 (0.42) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10568435 0.79 ATAD2 (0.41) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL9832061 0.77 PDE3B (0.49) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10566029 0.77 ATAD2 (0.39) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL9835825 0.77 PDK2 (0.50) ATAD2PDE3BPDE3APDE4APDE4B
Water SCHEMBL10470996 0.76 PDE3B (0.48) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10566915 0.76 ATAD2 (0.41) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10585407 0.76 KDM4E (0.55) PDE4APDE4BPDE4CPDE4DPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed