SCHEMBL1056743

SCHEMBL1056743

CC(=O)c1ccc(C)c(OS(=O)(=O)C(F)(F)F)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.43
CXCR2 P25025 2/20 0.35
CXCR1 P25024 1/20 0.35
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP2C19 P33261 2/20 0.31
NOTUM Q6P988 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
USP2 O75604 1/20 0.31
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23925994 0.83 TSHR (0.41) ALDH1A1KDM4EHSD17B10MAPTPDK2
SCHEMBL23250280 0.82 CXCR2 (0.35) HSD11B1CXCR2CXCR1NOTUM
SCHEMBL29863304 0.82 CXCR2 (0.35) HSD11B1CXCR2CXCR1NOTUM
SCHEMBL17205759 0.80 KDM4E (0.37) HSD11B1CXCR2CXCR1ALDH1A1HPGD
SCHEMBL27351302 0.77 HSD11B1 (0.56) HSD11B1CXCR2CXCR1ALDH1A1HPGD
SCHEMBL1748180 0.77 HSD11B1 (0.56) HSD11B1CXCR2CXCR1ALDH1A1HPGD
SCHEMBL8434832 0.77 HSD11B1 (0.44) HSD11B1CXCR2CXCR1ALDH1A1HPGD
SCHEMBL19330864 0.77 CFTR (0.38) HSD11B1CXCR2CXCR1ALDH1A1HPGD
SCHEMBL9275010 0.75 ALDH1A1 (0.38) ALDH1A1HPGDHSD17B10CYP2C19NOTUM
SCHEMBL7318290 0.75 MAPT (0.51) HSD11B1CXCR2CXCR1CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008725-A2 METAL-CATALYZED CARBON-FLUORINE BOND FORMATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2011-01-20 WO disclosed
US-20110015401-A1 Metal-Catalyzed Carbon-Fluorine Bond Formation MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2011-01-20 US disclosed
WO-2011008618-A1 METAL-CATALYZED CARBON-FLUORINE BOND FORMATION NATIONAL UNIVERSITY OF SINGAPORE (SG) 2011-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110015401-A1 Metal-Catalyzed Carbon-Fluorine Bond Formation FLI1, VGF, GMFG HSD11B1 3639/4885CXCR2 2378/4885CXCR1 2052/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.