SCHEMBL10567463

SCHEMBL10567463

Cc1cc(Cl)c2[nH]nc(-c3ccccc3)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.46
YTHDC1 Q96MU7 1/20 0.43
YTHDF2 Q9Y5A9 1/20 0.43
MAPT P10636 5/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 2/20 0.41
CRHR1 P34998 2/20 0.41
ALDH1A1 P00352 3/20 0.39
GFER P55789 1/20 0.39
ADORA1 P30542 3/20 0.39
ADORA2A P29274 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
KDM4E B2RXH2 3/20 0.38
MAPK10 P53779 2/20 0.38
ALPL P05186 1/20 0.38
GAA P10253 1/20 0.38
IDO1 P14902 1/20 0.38
TTK P33981 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10564706 0.88 CRHR1 (0.46) HPGDMAPTL3MBTL1LMNACRHR1
SCHEMBL10568473 0.83 MEN1 (0.47) HPGDMAPTLMNACRHR1ALDH1A1
SCHEMBL10568466 0.78 ALDH1A1 (0.43) HPGDLMNACRHR1ALDH1A1KDM4E
SCHEMBL10566728 0.75 MAPT (0.39) MAPTL3MBTL1LMNACRHR1ALDH1A1
SCHEMBL10571998 0.73 YTHDC1 (0.40) YTHDC1YTHDF2MEN1KMT2ARAB9A
SCHEMBL10569381 0.73 CYP2C19 (0.51) HPGDYTHDC1YTHDF2L3MBTL1ALDH1A1
SCHEMBL5358160 0.73 ALDH1A1 (0.46) HPGDYTHDC1YTHDF2MAPTL3MBTL1
SCHEMBL10567327 0.72 YTHDC1 (0.41) HPGDYTHDC1YTHDF2L3MBTL1LMNA
SCHEMBL6851931 0.72 MAPT (0.40) MAPTL3MBTL1LMNACRHR1ALDH1A1
SCHEMBL10565223 0.72 CHEK1 (0.41) MAPTL3MBTL1LMNACRHR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833136-A ANTIINFLAMMATORY AGENTS BEECHAM GROUP P.L.C. (GB) 1989-05-23 US disclosed
EP-0239191-A2 Pyrazolo[4,3-b]pyridine derivatives, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1987-09-30 EP disclosed