SCHEMBL10568375

SCHEMBL10568375

COC(=O)c1c(S(=O)(=O)NC(=O)Nc2nc(C)cc(OC)n2)c2ccccc2n1C

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
GAA P10253 2/20 0.45
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PABPC1 P11940 1/20 0.39
EIF4H Q15056 1/20 0.39
CDK1 P06493 1/20 0.38
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.36
CASR P41180 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567289 0.93 ALDH1A1 (0.56) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10566127 0.93 SMN1; SMN2 (0.46) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10569523 0.87 GAA (0.51) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10974258 0.85 GAA (0.44) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10565455 0.83 GAA (0.43) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL11043791 0.79 GAA (0.49) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL11162591 0.79 GAA (0.46) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL9419172 0.78 GAA (0.52) KDM4EGAATSHRSMN1; SMN2CDK1
SCHEMBL11045447 0.78 GAA (0.40) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10565848 0.78 ALDH1A1 (0.45) KDM4EALDH1A1HPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4836846-A PRE/POST EMERGENCE; WEEDS, GRASSES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-06-06 US disclosed
US-4764610-A Herbicidal indole sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-08-16 US disclosed
EP-0070698-B1 HERBICIDAL INDOLE SULFONAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-11-13 EP disclosed
EP-0070698-A1 Herbicidal indole sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-01-26 EP disclosed