SCHEMBL10568467

SCHEMBL10568467

OC/C=C(/c1ccccc1)c1ncccn1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.52
CTNNB1 P35222 1/20 0.46
WNT3A P56704 1/20 0.46
CYP19A1 P11511 2/20 0.44
CYP11B2 P19099 2/20 0.44
TBXAS1 P24557 7/20 0.40
TBXA2R P21731 3/20 0.38
KMT2A Q03164 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10568471 1.00 TDP1 (0.52) TDP1CTNNB1WNT3ACYP19A1CYP11B2
SCHEMBL6421667 0.81 KMT2A (0.50) TDP1KMT2ACYP2D6
SCHEMBL6421671 0.81 KMT2A (0.50) TDP1KMT2ACYP2D6
SCHEMBL4630812 0.81 MTNR1A (0.48) TDP1CYP19A1CYP11B2TBXAS1CHRNB2
SCHEMBL6419179 0.78 CYP19A1 (0.55) CYP19A1CYP11B2TBXAS1TBXA2RKMT2A
SCHEMBL6419131 0.78 CYP19A1 (0.55) CYP19A1CYP11B2TBXAS1TBXA2RKMT2A
SCHEMBL28961178 0.74 CYP19A1 (0.66) TDP1CTNNB1WNT3ACYP19A1CYP11B2
SCHEMBL8699447 0.74 TBXAS1 (0.68) TBXAS1TBXA2R
SCHEMBL8699446 0.74 TBXAS1 (0.68) TBXAS1TBXA2R
SCHEMBL10566764 0.73 TDP1 (0.52) TDP1CTNNB1WNT3ACYP19A1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831034-A 4-benzylpiperazines useful as neuroleptics RHONE-POULENC SANTE (FR) 1989-05-16 US disclosed