SCHEMBL10568512

SCHEMBL10568512

CS(=O)(=O)Nc1ccc(CS(=O)(=O)Oc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.65
PGR P06401 2/20 0.59
HPGD P15428 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
AR P10275 2/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
KEAP1 Q14145 1/20 0.53
HTT P42858 2/20 0.53
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
ADRB3 P13945 1/20 0.50
NR3C2 P08235 4/20 0.48
RORA P35398 1/20 0.46
RORC P51449 1/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14607550 0.81 KMT2A (0.69) KMT2APGRARHTTLMNA
Hydrochloric Acid SCHEMBL10465859 0.80 KMT2A (0.67) KMT2APGRARHTTLMNA
Phenyl Phenylmethanesulfonate SCHEMBL6912876 0.80 KMT2A (1.00) KMT2APGRHPGDARHTT
Phenyl Phenylmethanesulfonate SCHEMBL27917341 0.78 KMT2A (0.96) KMT2APGRHPGDARHTT
SCHEMBL9479731 0.76 KMT2A (0.71) KMT2APGRHPGDSMN1; SMN2AR
SCHEMBL10571949 0.76 KMT2A (0.76) KMT2APGRSMN1; SMN2NPC1RAB9A
SCHEMBL28790351 0.75 HPGD (0.85) PGRHPGDSMN1; SMN2ARNPC1
SCHEMBL28015271 0.75 PGR (1.00) PGRHPGDSMN1; SMN2ARNPC1
Hydrochloric Acid SCHEMBL10466655 0.74 KMT2A (0.73) KMT2APGRSMN1; SMN2NPC1RAB9A
SCHEMBL22187191 0.73 CA2 (0.57) KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4855314-A VASOCONTRICTORS, TREATMENT OF MIGRAINES, 3-(AMINO-ETHYL)-5-(PHENYL(ALKYL)-CARBONYL OR SULFONYL-AMINOALKYL SUBSTITUTED GLAXO GROUP LIMITED (GB) 1989-08-08 US disclosed
EP-0240096-A1 Indole derivatives having a selective vasoconstrictor activity GLAXO GROUP LIMITED (GB) 1987-10-07 EP disclosed