SCHEMBL10568585

SCHEMBL10568585

COc1ccc(C2C3=C(CCCC3)CCN2C(C)=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
POLB P06746 2/20 0.42
LHCGR P22888 6/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
RECQL P46063 1/20 0.41
TP53 P04637 2/20 0.41
ABCB1 P08183 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HHAT Q5VTY9 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545035 0.81 CYP3A4 (0.48) SMN1; SMN2MEN1KMT2AGAA
SCHEMBL11447599 0.73 CYP3A4 (0.46) TSHRSMN1; SMN2RECQLKDM4EMAPT
SCHEMBL9151971 0.73 CYP2D6 (0.61) SMN1; SMN2MEN1KMT2AGAA
SCHEMBL11757293 0.73 CYP2D6 (0.61) SMN1; SMN2MEN1KMT2AGAA
SCHEMBL11465395 0.72 CYP3A4 (0.45) TSHRSMN1; SMN2RECQLMEN1KMT2A
SCHEMBL11755929 0.70 HSD11B1 (0.46) SMN1; SMN2TP53
SCHEMBL19427415 0.69 CYP3A4 (0.49) SMN1; SMN2TP53MEN1KMT2AKDM4E
SCHEMBL985851 0.67 MTNR1B (0.56) TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL998666 0.67 ABCG2 (0.57) SMN1; SMN2TP53ABCB1ABCG2KMT2A
SCHEMBL23397304 0.66 ALDH1A1 (0.51) POLBMEN1KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4857648-A Isoquinoline derivatives HOFFMANN-LA ROCHE INC. (US) 1989-08-15 US claimed