SCHEMBL10573299

SCHEMBL10573299

NS(=O)(=O)c1cc2cc3c(cc2[nH]1)OCO3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 1.00
AKR1B1 P15121 1/20 0.54
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
GAA P10253 1/20 0.35
KIF11 P52732 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11016994 0.77 CA2 (0.62) CA2AKR1B1KDM4EALDH1A1GAA
SCHEMBL10573479 0.73 CA2 (0.66) CA2CA12CA9
SCHEMBL4450283 0.71 AKR1B1 (1.00) CA2AKR1B1
SCHEMBL16821915 0.70 CA2 (0.54) CA2AKR1B1KDM4EALDH1A1RAB9A
SCHEMBL7493903 0.69 CA2 (0.53) CA2AKR1B1KDM4EALDH1A1GAA
SCHEMBL2400125 0.68 GPR35 (0.56) CA2AKR1B1KDM4EALDH1A1RAB9A
SCHEMBL13850474 0.68 CA2 (0.51) CA2AKR1B1KDM4EALDH1A1GAA
SCHEMBL30817138 0.68 GPR35 (0.56) CA2AKR1B1KDM4EALDH1A1RAB9A
SCHEMBL10573193 0.68 CA2 (0.62) CA2CA12CA9KDM4EALDH1A1
SCHEMBL8980508 0.67 AKR1B1 (0.51) CA2AKR1B1CA12CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4840963-A FOR GLAUCOMA MERCK & CO., INC. (US) 1989-06-20 US disclosed
EP-0155214-A2 2-sulfamoyl-1H-indole derivatives for the treatment of elevated intraocular pressure MERCK & CO. INC. (US) 1985-09-18 EP disclosed