SCHEMBL10577331

SCHEMBL10577331

C=CCn1c(=O)c2cnccc2n(CC=C)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 4/20 0.44
ADORA2A P29274 3/20 0.44
CYP3A4 P08684 2/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ROCK2 O75116 1/20 0.42
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CMA1 P23946 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAOA P21397 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523462 0.78 GAA (0.53) ADORA2BADORA2ACYP3A4KMT2AGAA
SCHEMBL4551429 0.76 KDM5A (0.48) ADORA2BADORA2AKMT2AROCK2CMA1
SCHEMBL18901219 0.74 ROCK2 (0.56) KMT2AGAAKDM4EMEN1LMNA
SCHEMBL16377261 0.72 ROCK2 (0.63) KMT2AKDM4EMEN1LMNAHTT
SCHEMBL29507760 0.69 CYP3A4 (0.62) CYP3A4KMT2AGAAKDM4ELMNA
SCHEMBL6695468 0.69 CYP3A4 (0.62) CYP3A4KMT2AGAAKDM4ELMNA
SCHEMBL3361253 0.69 MAOA (0.50) KMT2AGAAKDM4EMEN1LMNA
SCHEMBL16377262 0.69 ROCK2 (0.64) KMT2AKDM4EMEN1LMNAHTT
SCHEMBL11498958 0.69 MEN1 (0.48) KMT2AGAAKDM4EMEN1LMNA
SCHEMBL9778174 0.65 CYP3A4 (0.50) ADORA2BADORA2ACYP3A4KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4808618-A ANTIALLERGENS NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1989-02-28 US disclosed