SCHEMBL8523462

SCHEMBL8523462

C=CCn1c(=O)c2ccccc2n(CC=C)c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
PLK1 P53350 1/20 0.53
APOBEC3G Q9HC16 1/20 0.53
KDM4E B2RXH2 3/20 0.50
MAPT P10636 2/20 0.50
CYP3A4 P08684 1/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
LMNA P02545 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4C Q9H3R0 1/20 0.46
ALPL P05186 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14692503 0.85 ADORA2B (0.53) GAAPLK1APOBEC3GKDM4ECYP3A4
SCHEMBL29507760 0.85 CYP3A4 (0.62) GAAPLK1APOBEC3GKDM4ECYP3A4
SCHEMBL6695468 0.85 CYP3A4 (0.62) GAAPLK1APOBEC3GKDM4ECYP3A4
SCHEMBL6454733 0.84 CNR2 (0.56) PLK1APOBEC3GKDM4EMAPTALDH1A1
SCHEMBL9709253 0.80 ALDH1A1 (0.58) GAAPLK1APOBEC3GMEN1KMT2A
SCHEMBL30493502 0.80 ALDH1A1 (0.58) GAAPLK1APOBEC3GMEN1KMT2A
SCHEMBL146503 0.79 CYP1A2 (0.56) GAAAPOBEC3GKDM4EMAPTCYP3A4
SCHEMBL10577331 0.78 ADORA2B (0.44) GAAPLK1APOBEC3GKDM4EMAPT
SCHEMBL24031109 0.78 HDAC1 (0.77) KDM4EMAPTSMN1; SMN2MAPK1L3MBTL1
SCHEMBL4593193 0.75 HSP90AA1 (0.46) GAAPLK1APOBEC3GKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999002990-A1 COMBINATORIAL PROCESS FOR PREPARING FUSED SUBSTITUTED PYRIMIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1999-01-21 WO disclosed