SCHEMBL10577832

SCHEMBL10577832

Cn1ccnc1N1CCN(CC(=O)c2ccc(NS(C)(=O)=O)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.43
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 3/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 2/20 0.39
POLB P06746 2/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ADRB2 P07550 2/20 0.39
ADRB1 P08588 2/20 0.39
ADRB3 P13945 2/20 0.39
KCNH2 Q12809 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10579790 0.81 ADRB2 (0.47) GRIN2BKDM4EGAAMEN1KMT2A
SCHEMBL10359739 0.81 POLB (0.57) GRIN2BALDH1A1TDP1POLBGAA
SCHEMBL10677172 0.81 JAK2 (0.47) GRIN2BALDH1A1SMN1; SMN2POLBGAA
SCHEMBL9513736 0.80 POLB (0.49) GRIN2BALDH1A1KDM4ETSHRHTT
SCHEMBL9514727 0.78 POLB (0.43) GRIN2BALDH1A1KDM4ETSHRHTT
SCHEMBL9514777 0.77 CA1 (0.46) GRIN2BALDH1A1KDM4ETSHRHTT
SCHEMBL10581142 0.77 GRIN2B (0.42) GRIN2BALDH1A1KDM4ETSHRHTT
SCHEMBL9515021 0.77 NAMPT (0.51) GRIN2BALDH1A1KDM4ETSHRHTT
SCHEMBL10646175 0.76 ALDH1A1 (0.56) GRIN2BALDH1A1TSHRHTTMEN1
SCHEMBL9625464 0.76 ALDH1A1 (0.56) GRIN2BALDH1A1TSHRHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4806536-A Piperazinyl-substituted pyridine and imidazole anti-arrhythmic agents PFIZER, INC. (US) 1989-02-21 US disclosed
EP-0233051-A2 Antiarrhythmic Agents Pfizer Limited (GB) 1987-08-19 EP disclosed