SCHEMBL10600409

SCHEMBL10600409

CC[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)C(C#CCl)C[C@]4(C)C3=CC[C@@]21C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.43
CYP19A1 P11511 8/20 0.38
AR P10275 3/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
KCNH2 Q12809 1/20 0.34
ESR1 P03372 1/20 0.33
CHRM2 P08172 1/20 0.33
ACHE P22303 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CYP2C19 P33261 1/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
STS P08842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7189243 0.85 NR3C1 (0.47) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL4826656 0.80 NR3C1 (0.64) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL9470387 0.73 ESR1 (0.46) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL14571254 0.72 NR3C1 (0.64) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL8242650 0.72 NR3C1 (0.64) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL10530695 0.71 NR3C1 (0.55) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL10413728 0.69 NR3C1 (0.58) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL11321023 0.68 NFKB1 (0.41) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL4978357 0.68 NR3C1 (0.61) NR3C1CYP19A1ARPGRNR3C2
SCHEMBL4978346 0.68 NR3C1 (0.61) NR3C1CYP19A1ARPGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0181442-B1 PROCESS FOR THE PREPARATION OF PREGNANE DERIVATIVE SCHERING AKTIENGESELLSCHAFT (DE) 1989-07-12 EP disclosed
US-4708823-A 17 α-chloroethynyl pregnane derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1987-11-24 US disclosed