SCHEMBL10601002

SCHEMBL10601002

FC(F)Oc1ccc2cnn(SC(F)(Cl)Cl)c2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
RORC P51449 1/20 0.35
CYP3A4 P08684 2/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
ABL1 P00519 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2E1 P05181 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2B6 P20813 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGDS O60760 1/20 0.32
LRRK2 Q5S007 6/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10603126 0.91 NR3C1 (0.35) CYP17A1CYP2C9CYP2C19CYP3A4ABL1
SCHEMBL10602397 0.88 ATP4A (0.35) HTR2AHTR2CHTR2BATP4AATP4B
SCHEMBL10597717 0.86 PDE10A (0.38) CYP2C9CYP3A4CYP1A2ALDH1A1GAA
SCHEMBL10599937 0.81 CYP17A1 (0.40) CYP17A1CYP2C9CYP2C19HTR2AHTR2C
SCHEMBL10619578 0.80 PDE10A (0.37) CYP2C9CYP3A4CYP1A2ALDH1A1GAA
SCHEMBL10602392 0.79 ATP4A (0.33) ATP4AATP4B
SCHEMBL10601241 0.77 GPR3 (0.36) CYP2C9CYP3A4CYP1A2GAACACNA1H
SCHEMBL10621858 0.76 PDE10A (0.39) CYP2C9CYP3A4CYP1A2ALDH1A1GAA
SCHEMBL10598423 0.76 KCNH2 (0.30)
SCHEMBL10603073 0.75 KCNH2 (0.38) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778511-A FOR PLANTS AND MATERIALS BAYER AKTIENGESELLSCHAFT (DE) 1988-10-18 US claimed
EP-0195238-B1 N-SULPHENYLIZED INDAZOLES CONTAINING FLUORINE, PROCESS FOR THEIR PREPARATION AND THEIR USE BAYER AG (DE) 1989-03-29 EP disclosed
US-4778511-A FOR PLANTS AND MATERIALS BAYER AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0195238-A1 N-sulphenylized indazoles containing fluorine, process for their preparation and their use BAYER AG (DE) 1986-09-24 EP disclosed