SCHEMBL15061997

SCHEMBL15061997

CC(=O)N1CCC(Oc2ccccc2C)CC1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.59
KMT2A Q03164 3/20 0.55
IKBKB O14920 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
CHUK O15111 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SCD O00767 1/20 0.48
NAMPT P43490 1/20 0.47
MEN1 O00255 1/20 0.46
RBP4 P02753 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9903544 0.88 EPHX2 (0.62) EPHX2KMT2ANPC1RAB9ASCD
SCHEMBL9013887 0.84 IKBKB (0.49) EPHX2KMT2AIKBKBCHUKNAMPT
SCHEMBL30352887 0.83 IKBKB (0.47) EPHX2IKBKBTDP1CHUKSCD
SCHEMBL28278842 0.82 EPHX2 (0.57) EPHX2KMT2ANPC1RAB9ASCD
SCHEMBL17559489 0.82 IKBKB (0.51) EPHX2IKBKBTDP1CHUKNAMPT
SCHEMBL21765007 0.82 KDM1A (0.57) EPHX2KMT2A
SCHEMBL10608977 0.81 EPHX2 (0.56) EPHX2KMT2ANPC1RAB9ASCD
SCHEMBL17955461 0.81 RBP4 (0.67) EPHX2IKBKBCHUKSCDNAMPT
SCHEMBL31202927 0.80 IKBKB (0.47) KMT2AIKBKBTDP1CHUKRAB9A
SCHEMBL13536484 0.80 EPHX2 (0.55) EPHX2KMT2ANPC1RAB9ASCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013091773-A1 TETRAAZA-CYCLOPENTA[A]INDENYL AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS MERCK PATENT GMBH (DE) 2013-06-27 WO disclosed
EP-2607364-A1 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators Ares Trading S.A. (CH) 2013-06-26 EP disclosed