SCHEMBL10609477

SCHEMBL10609477

O=c1cnc2[nH]cnc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
GDA Q9Y2T3 1/20 0.41
ALDH1A1 P00352 6/20 0.40
ADORA2B P29275 5/20 0.40
ADORA2A P29274 4/20 0.40
KDM4E B2RXH2 4/20 0.40
LMNA P02545 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GLA P06280 1/20 0.40
PMP22 Q01453 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
TSHR P16473 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
XDH P47989 1/20 0.39
RAB9A P51151 1/20 0.39
BLM P54132 1/20 0.39
ABL1 P00519 1/20 0.37
RIN1 Q13671 1/20 0.37
MAPKAPK2 P49137 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6379644 0.77 ALDH1A1 (0.53) ACHEGDAALDH1A1ADORA2AKDM4E
SCHEMBL6904582 0.77 ACHE (0.50) ACHEGDAALDH1A1ADORA2BADORA2A
SCHEMBL22487918 0.70 KDM4E (0.39) ALDH1A1KDM4ELMNAHSD17B10GLA
SCHEMBL20830320 0.70 ALDH1A1 (0.42) ALDH1A1KDM4ELMNAHSD17B10GLA
SCHEMBL1257032 0.67 MAPKAPK2 (0.51) ALDH1A1KDM4ESMN1; SMN2XDHRAB9A
SCHEMBL31156527 0.67 MAPKAPK2 (0.51) ALDH1A1KDM4ESMN1; SMN2XDHRAB9A
SCHEMBL6325739 0.67 ACHE (0.39) ACHEGDAADORA2BADORA2ALMNA
SCHEMBL20830317 0.67 ALDH1A1 (0.41) ACHEGDAALDH1A1ADORA2AKDM4E
SCHEMBL22487729 0.66 L3MBTL1 (0.39) ALDH1A1KDM4ELMNAHSD17B10GLA
SCHEMBL28588392 0.64 ALDH1A1 (0.65) ACHEGDAALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4670438-A Imidazo[4,5-c]pyridazine-3-ones, imidazo[4,5-d]pyridazine-4-ones, imidazo[4,]pyrazin-5-ones, purin-2-ones, purin-6-ones, and purin-2,6-diones useful as hypotensive or cardiotonic agents DR. KARL THOMAE GMBH (DE) 1987-06-02 US claimed
EP-0130461-A2 Imidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-01-09 EP claimed
US-4766130-A 2-phenyl-imidazopyridin-ones and also useful as cardiotonics and anti-hypertensives CELAMERCK GMBH & CO. KG (DE) 1988-08-23 US disclosed
US-4670438-A Imidazo[4,5-c]pyridazine-3-ones, imidazo[4,5-d]pyridazine-4-ones, imidazo[4,]pyrazin-5-ones, purin-2-ones, purin-6-ones, and purin-2,6-diones useful as hypotensive or cardiotonic agents DR. KARL THOMAE GMBH (DE) 1987-06-02 US disclosed
EP-0130461-A2 Imidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-01-09 EP disclosed