SCHEMBL10623972

SCHEMBL10623972

O=C1Cc2c(Cl)cccc2C(c2cccnc2)N1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
TRPM5 Q9NZQ8 2/20 0.38
MAPK1 P28482 2/20 0.36
GAA P10253 1/20 0.36
LDHA P00338 1/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
RECQL P46063 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
CHRNA7 P36544 1/20 0.35
CYP19A1 P11511 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10622394 0.78 SMN1; SMN2 (0.58) CHRNB2CHRNA4MAPK1GAAMAPT
SCHEMBL10625325 0.73 CYP3A4 (0.46) CHRNB2CHRNA4MAPTKMT2ASMN1; SMN2
SCHEMBL10626570 0.70 KMT2A (0.49) GAAKDM4EKMT2ACRHBPCRHR2
SCHEMBL7898965 0.70 MEN1 (0.46) CHRNB2CHRNA4TRPM5MAPK1GAA
SCHEMBL21261501 0.69 CYP19A1 (0.46) CHRNB2CHRNA4MAPK1GAAMAPT
Hydrochloric Acid SCHEMBL10626522 0.68 CYP11B2 (0.35) CHRNB2CHRNA4CHRNA7CYP19A1CYP11B1
SCHEMBL156842 0.67 CHRNB2 (0.56) CHRNB2CHRNA4MAPK1MAPTKDM4E
SCHEMBL4991736 0.67 CYP2A6 (0.45) CHRNB2CHRNA4MAPK1GAAKDM4E
SCHEMBL10622377 0.66 KMT2A (0.40) GAAKDM4EMEN1RAB9AKMT2A
SCHEMBL10624676 0.66 KMT2A (0.45) CHRNB2CHRNA4GAAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183369-A2 Dihydroisoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1986-06-04 EP claimed
US-4745115-A ANTIALLERGENS, RHEUMATIC DISEASES BEECHAM GROUP P.L.C. (GB) 1988-05-17 US disclosed
EP-0183369-A2 Dihydroisoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1986-06-04 EP disclosed