SCHEMBL10626

SCHEMBL10626

NC(=O)CCCc1ccc(-c2ccc(OCCCN3CCOCC3)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.63
HRH2 P25021 1/20 0.58
HRH1 P35367 1/20 0.58
MAPK1 P28482 2/20 0.55
ALDH1A1 P00352 1/20 0.55
CYP1A2 P05177 1/20 0.55
CHRM2 P08172 1/20 0.55
CHRM1 P11229 1/20 0.55
HTR2A P28223 1/20 0.55
SCN1A P35498 1/20 0.55
HTR2B P41595 1/20 0.55
KCNH2 Q12809 1/20 0.55
SCN2A Q99250 1/20 0.55
SIGMAR1 Q99720 1/20 0.55
SCN3A Q9NY46 1/20 0.55
USP2 O75604 1/20 0.54
LMNA P02545 1/20 0.54
EPHX2 P34913 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377 0.95 NPC1 (0.58) HRH3HRH2HRH1ALDH1A1LMNA
SCHEMBL10637 0.88 HRH3 (0.76) HRH3HRH1KCNH2
SCHEMBL27896953 0.83 HRH3 (0.76) HRH3HRH2HRH1MAPK1ALDH1A1
SCHEMBL10132932 0.81 EPHX2 (0.63) HRH3HRH2HRH1ALDH1A1EPHX2
SCHEMBL15577570 0.81 MEN1 (0.54) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL23963137 0.80 HRH3 (0.67) HRH3HRH2HRH1MAPK1ALDH1A1
SCHEMBL14714478 0.79 HRH3 (0.77) HRH3HRH2HRH1MAPK1ALDH1A1
SCHEMBL5306939 0.79 HDAC1 (0.57) ALDH1A1LMNAEPHX2
SCHEMBL29973108 0.79 HRH3 (0.69) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL14724514 0.79 HRH3 (0.71) HRH3HRH2HRH1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488489-A2 C-LINKED HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS Pfizer Inc. (US) 2012-08-22 EP disclosed
WO-2011045703-A2 C-LINKED HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS PFIZER INC. (US) 2011-04-21 WO disclosed