SCHEMBL10377

SCHEMBL10377

NC(=O)CCCc1ccc(-c2ccc(OCCN3CCOCC3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
HRH3 Q9Y5N1 8/20 0.57
LTA4H P09960 1/20 0.54
GAA P10253 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
HRH2 P25021 1/20 0.52
HRH1 P35367 1/20 0.52
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
THRB P10828 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10626 0.95 HRH3 (0.63) HRH3ALDH1A1HRH2HRH1LMNA
SCHEMBL5306939 0.84 HDAC1 (0.57) LTA4HGAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL10637 0.83 HRH3 (0.76) HRH3HRH1
SCHEMBL1395845 0.83 LTA4H (0.61) NPC1RAB9ALTA4HGAASMN1; SMN2
SCHEMBL31427171 0.82 LTA4H (0.64) NPC1RAB9ALTA4HGAASMN1; SMN2
SCHEMBL874263 0.81 ALDH1A1 (0.64) NPC1RAB9AHRH3LTA4HGAA
SCHEMBL28502559 0.81 NPC1 (0.67) NPC1RAB9AHRH3LTA4HGAA
SCHEMBL874183 0.80 LTA4H (0.61) NPC1RAB9AHRH3LTA4HCA12
SCHEMBL10132861 0.80 NPC1 (0.63) NPC1RAB9AHRH3LTA4HGAA
SCHEMBL873542 0.79 ALDH1A1 (0.74) NPC1RAB9AHRH3LTA4HGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488489-A2 C-LINKED HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS Pfizer Inc. (US) 2012-08-22 EP disclosed
WO-2011045703-A2 C-LINKED HYDROXAMIC ACID DERIVATIVES USEFUL AS ANTIBACTERIAL AGENTS PFIZER INC. (US) 2011-04-21 WO disclosed