SCHEMBL15577570

SCHEMBL15577570

NC(=O)C(O)c1ccc(CCCCc2ccc(OCCCN3CCOCC3)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
KMT2A Q03164 1/20 0.54
HRH3 Q9Y5N1 11/20 0.52
MAPK1 P28482 2/20 0.52
ALDH1A1 P00352 2/20 0.52
CYP1A2 P05177 1/20 0.52
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
HTR2A P28223 1/20 0.52
SCN1A P35498 1/20 0.52
HTR2B P41595 1/20 0.52
KCNH2 Q12809 1/20 0.52
SCN2A Q99250 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
SCN3A Q9NY46 1/20 0.52
USP2 O75604 1/20 0.51
LMNA P02545 1/20 0.51
EPHX2 P34913 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10626 0.81 HRH3 (0.63) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL15522497 0.78 EPHX2 (0.60) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL15522535 0.78 EPHX2 (0.66) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL23963137 0.77 HRH3 (0.67) KMT2AHRH3MAPK1ALDH1A1CYP1A2
SCHEMBL15581514 0.77 EPHX2 (0.64) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL10377 0.76 NPC1 (0.58) NPC1RAB9AKMT2AHRH3ALDH1A1
SCHEMBL29973108 0.76 HRH3 (0.69) KMT2AHRH3MAPK1ALDH1A1CYP1A2
SCHEMBL10625 0.76 HRH3 (0.61) MEN1NPC1RAB9AKMT2AHRH3
SCHEMBL874183 0.75 LTA4H (0.61) NPC1RAB9AKMT2AHRH3MAPK1
SCHEMBL23291288 0.75 EPHX2 (0.60) HRH3MAPK1ALDH1A1CYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014041424-A1 HISTONE DEACETYLASE INHIBITORS FOR ENHANCING ACTIVITY OF ANTIFUNGAL AGENTS METHYLGENE INC. (CA) 2014-03-20 WO disclosed