SCHEMBL10633765

SCHEMBL10633765

CC(C)c1cccc(C(C)(C)c2ccccc2)c1C(C)(C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
CYP3A4 P08684 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2C19 P33261 1/20 0.37
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
GABRA1 P14867 3/20 0.36
LMNA P02545 3/20 0.36
GABRB2 P47870 2/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
FAAH O00519 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
GABRB1 P18505 1/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29932235 0.89 CYP3A4 (0.42) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
Hydrogen Peroxide SCHEMBL28707558 0.87 CYP3A4 (0.45) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
SCHEMBL6546769 0.85 CRHBP (0.43) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
Hydrogen Peroxide SCHEMBL9064510 0.83 CRHBP (0.46) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
SCHEMBL10775084 0.81 GABRA1 (0.53) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
SCHEMBL985925 0.81 GABRA1 (0.52) CRHBPCRHR2CYP3A4ALDH1A1ESR1
SCHEMBL28101263 0.78 NR3C2 (0.40) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
SCHEMBL15105312 0.78 ALDH1A1 (0.39) CRHBPCRHR2CYP3A4ALDH1A1ESR1
SCHEMBL11829651 0.77 CYP3A4 (0.36) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19
SCHEMBL25137938 0.76 CYP3A4 (0.36) CRHBPCRHR2CYP3A4ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4752641-A POLYFUNCTIONAL MALEIMIDE, ALKENYLPHENOLS OR ALKENYLPHENOL ETHERS, AND ALLYL ESTER OF POLYVALENT CARBOXYLIC ACID OR CYANURIC OR ISOCYANURIC ACID HITACHI, LTD. (JP) 1988-06-21 US disclosed