SCHEMBL10640211

SCHEMBL10640211

COC(=O)/C=C/C=C/c1ccccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.41
CAPN1 P07384 2/20 0.41
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
GAA P10253 2/20 0.40
ABCB1 P08183 2/20 0.40
F2R P25116 1/20 0.40
TFEB P19484 1/20 0.40
ALDH1A1 P00352 5/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.37
TSHR P16473 1/20 0.37
POLB P06746 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
TYR P14679 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10640215 1.00 NFE2L2 (0.41) NFE2L2CAPN1CTSLCTSBGAA
SCHEMBL4281638 0.89 ALDH1A1 (0.46) NFE2L2GAAF2RTFEBALDH1A1
SCHEMBL4281639 0.89 ALDH1A1 (0.46) NFE2L2GAAF2RTFEBALDH1A1
SCHEMBL1399174 0.85 GAA (0.48) CAPN1CTSLCTSBGAAALDH1A1
SCHEMBL1399096 0.85 GAA (0.48) CAPN1CTSLCTSBGAAALDH1A1
SCHEMBL1399130 0.81 CA1 (0.43) GAAF2RALDH1A1L3MBTL1KDM4E
SCHEMBL1399132 0.81 CA1 (0.43) GAAF2RALDH1A1L3MBTL1KDM4E
SCHEMBL7134613 0.76 GAA (0.36) GAAF2RALDH1A1L3MBTL1POLB
SCHEMBL7134611 0.76 GAA (0.36) GAAF2RALDH1A1L3MBTL1POLB
SCHEMBL11554418 0.75 NFE2L2 (0.54) NFE2L2GAAF2RTFEBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153720-B1 SPERGUALIN-RELATED COMPOUNDS HAVING A PHENYLENE GROUP, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1988-11-09 EP disclosed
US-4556735-A BACTERICIDE, ANTITUMOR AGENT ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1985-12-03 US disclosed
EP-0153720-A2 Spergualin-related compounds having a phenylene group, a process for their preparation and their use as medicaments MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1985-09-04 EP disclosed