SCHEMBL10643134

SCHEMBL10643134

CC(CC(N)(O)c1cccc(Cl)c1)OC(N)=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 3/20 0.44
SCN9A Q15858 3/20 0.44
KIF11 P52732 2/20 0.40
PKM P14618 1/20 0.39
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
RAB9A P51151 1/20 0.38
OGG1 O15527 1/20 0.37
PARP1 P09874 1/20 0.36
CCR6 P51684 1/20 0.36
KCNH2 Q12809 1/20 0.36
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
PNMT P11086 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27363440 0.80 SCN5A (0.43) SCN5ASCN9AKIF11PKMPNMT
SCHEMBL10643127 0.72 SCN5A (0.48) SCN5ASCN9AKIF11PKMPARP1
SCHEMBL9015877 0.72 SCN5A (0.49) SCN5ASCN9AKIF11PKMPNMT
SCHEMBL19731492 0.70 CYP19A1 (0.45) SCN5ASCN9AKIF11PARP1CCR6
SCHEMBL30914002 0.68 KIF11 (0.42) SCN5ASCN9AKIF11PKMHPGD
SCHEMBL30913940 0.68 KIF11 (0.42) SCN5ASCN9AKIF11PKMHPGD
SCHEMBL30914073 0.68 KIF11 (0.42) SCN5ASCN9AKIF11PKMHPGD
SCHEMBL24729465 0.68 ADRA1D (0.47) HPGDALOX15OGG1PARP1
SCHEMBL17844752 0.68 ADRA1D (0.47) HPGDALOX15OGG1PARP1
SCHEMBL29927069 0.68 ADRA1D (0.47) HPGDALOX15OGG1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278621-A1 Substituted amine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-08-17 EP disclosed