SCHEMBL10646367

SCHEMBL10646367

CS(=O)(=O)Nc1ccc(C(=O)O)cc1.[NaH]

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.57
PTGS2 P35354 2/20 0.57
RECQL P46063 1/20 0.57
KEAP1 Q14145 1/20 0.57
KMT2A Q03164 2/20 0.53
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA9 Q16790 2/20 0.53
KDM4E B2RXH2 2/20 0.53
LMNA P02545 2/20 0.53
NR3C2 P08235 1/20 0.53
HTT P42858 2/20 0.52
ALDH1A1 P00352 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
PGR P06401 1/20 0.50
GFER P55789 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118340 0.98 KEAP1 (0.59) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL2044935 0.92 KIF11 (0.59) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL3555520 0.88 KDM4E (0.59) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL10417625 0.86 HPGD (0.56) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL3019804 0.85 PTPN11 (0.50) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL13157249 0.85 NPC1 (0.59) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL3555970 0.84 NPC1 (0.61) HPGDRECQLLMNASMN1; SMN2PGR
SCHEMBL4624606 0.82 HPGD (0.64) HPGDPTGS2RECQLKEAP1KMT2A
SCHEMBL7745099 0.82 HPGD (0.59) HPGDPTGS2RECQLKEAP1CA12
SCHEMBL27183018 0.82 PTPRB (0.57) KMT2ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0158775-B1 SUBSTITUTED SULFONAMIDOBENZAMIDES, ANTIARRYTHMIC AGENTS AND COMPOSITIONS THEREOF SCHERING AKTIENGESELLSCHAFT (DE) 1988-04-20 EP disclosed
US-4629739-A Substituted sulfonamidobenzamides and method of treating arrhythmias SCHERING A.G. (DE) 1986-12-16 US disclosed
EP-0158775-A1 Substituted sulfonamidobenzamides, antiarrythmic agents and compositions thereof SCHERING AKTIENGESELLSCHAFT (DE) 1985-10-23 EP disclosed
US-4544654-A Substituted sulfonamidobenzamides, antiarrhythmic agents and compositions thereof SCHERING A.G. (DE) 1985-10-01 US disclosed