SCHEMBL10650189

SCHEMBL10650189

Cc1nc(CCn2cnc3c2c(=O)n(C)c(=O)n3C)no1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
ADORA2B P29275 10/20 0.58
LMNA P02545 2/20 0.58
MAPT P10636 1/20 0.58
TSHR P16473 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
MAPK1 P28482 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10649350 0.93 ADORA2B (0.61) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10649455 0.92 ADORA2B (0.62) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10649548 0.91 ADORA2B (0.60) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL6438430 0.90 ADORA2B (0.56) ALDH1A1ADORA2BLMNAMAPTSMN1; SMN2
SCHEMBL10654724 0.86 ADORA2B (0.60) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10652809 0.85 ALDH1A1 (0.56) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10651743 0.84 ADORA2B (0.61) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10651816 0.83 ADORA2B (0.63) ALDH1A1ADORA2BLMNAMAPTTSHR
SCHEMBL10649753 0.83 SMN1; SMN2 (0.63) ALDH1A1ADORA2BLMNASMN1; SMN2RXFP1
SCHEMBL10650788 0.82 ADORA2B (0.64) ALDH1A1ADORA2BLMNAMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0089028-B1 THEOPHYLLIN DERIVATIVES, AND PROCESS FOR THEIR PREPARATION CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1988-05-25 EP claimed
EP-0089028-B1 THEOPHYLLIN DERIVATIVES, AND PROCESS FOR THEIR PREPARATION CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1988-05-25 EP disclosed
US-4565817-A ANTITUSSIVE AGENTS CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA R.T. (HU) 1986-01-21 US disclosed
EP-0089028-A1 Theophyllin derivatives, and process for their preparation CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1983-09-21 EP disclosed