SCHEMBL10651304

SCHEMBL10651304

CCOC(=S)Cc1ccc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 1/20 0.46
XBP1 P17861 1/20 0.46
HPD P32754 1/20 0.44
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPK1 P28482 3/20 0.43
GAA P10253 1/20 0.42
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10652415 0.86 CYP3A4 (0.48) ALDH1A1KDM4ECYP3A4CYP2C9XBP1
SCHEMBL30695843 0.86 CYP3A4 (0.48) ALDH1A1KDM4ECYP3A4CYP2C9XBP1
SCHEMBL10653936 0.83 MAPT (0.49) ALDH1A1CYP3A4MAPTLMNAMEN1
SCHEMBL3601604 0.82 CYP1A2 (0.58) ALDH1A1KDM4EMAPTLMNAMEN1
SCHEMBL10511891 0.81 CYP1A2 (0.47) ALDH1A1KDM4ECYP3A4HPDMAPT
SCHEMBL10511895 0.81 CYP1A2 (0.47) ALDH1A1KDM4ECYP3A4HPDMAPT
SCHEMBL10652124 0.81 MEN1 (0.44) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL10650486 0.80 MAPT (0.53) ALDH1A1KDM4ECYP3A4MAPTLMNA
SCHEMBL13678600 0.79 MAPK1 (0.53) ALDH1A1KDM4ECYP3A4HPDMAPT
SCHEMBL27956774 0.79 HPD (0.48) ALDH1A1KDM4ECYP3A4CYP2C9XBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4755509-A Heterocyclic aldose reductase inhibitors and methods of using them Carbipem (FR) 1988-07-05 US disclosed