SCHEMBL10653530

SCHEMBL10653530

COC(=O)CCC/C=C\c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.51
HDAC1 Q13547 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
PAM P19021 1/20 0.47
LMNA P02545 1/20 0.46
PPARG P37231 1/20 0.45
TBXAS1 P24557 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
MAOB P27338 1/20 0.44
TSHR P16473 1/20 0.44
CYP4F2 P78329 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29016750 1.00 AKT1 (0.51) AKT1HDAC1HDAC8HDAC3HDAC4
SCHEMBL22146948 0.94 HDAC1 (0.52) AKT1HDAC1HDAC8HDAC3HDAC4
SCHEMBL17490828 0.94 HDAC1 (0.52) AKT1HDAC1HDAC8HDAC3HDAC4
SCHEMBL19452350 0.90 AKT1 (0.62) AKT1HDAC1HDAC8HDAC3HDAC4
SCHEMBL7571411 0.90 AKT1 (0.62) AKT1HDAC1HDAC8HDAC3HDAC4
SCHEMBL9427247 0.84 GSK3B (0.55) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL9208139 0.84 GSK3B (0.55) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL29260522 0.84 PTGS2 (0.55) LMNAMAOBTSHRCYP4F2CYP4A11
SCHEMBL9427239 0.84 GSK3B (0.55) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL11647238 0.84 PAM (0.45) HDAC1HDAC8HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123543-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION AND USE AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1988-02-03 EP disclosed
US-4609744-A 4-oxo-benzopyran carboxylic acids MERCK FROSST CANADA INC. (CA) 1986-09-02 US disclosed
EP-0123543-A1 Leukotriene antagonists, their production and use and compositions containing them MERCK FROSST CANADA INC. (CA) 1984-10-31 EP disclosed