SCHEMBL10658124

SCHEMBL10658124

Cn1c(=S)sc2ncccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2A6 P11509 2/20 0.35
HTR3E A5X5Y0 2/20 0.35
HTR3B O95264 2/20 0.35
HTR3A P46098 2/20 0.35
HTR3D Q70Z44 2/20 0.35
HTR3C Q8WXA8 2/20 0.35
HTT P42858 1/20 0.35
RPS6KA5 O75582 1/20 0.34
PDK1 Q15118 1/20 0.33
PRNP P04156 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19152972 0.78 CYP2A6 (0.39) SMN1; SMN2CYP2A6HTTRPS6KA5PDK1
SCHEMBL230331 0.68 F12 (0.59) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL18237780 0.67 POLB (0.37) KDM4ECYP2A6POLBALDH1A1
Hydrochlorthiazide SCHEMBL9107872 0.66 F12 (0.42) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL2628342 0.65 ADORA3 (0.54) MAPTKDM4ENPC1SMN1; SMN2NFKB1
SCHEMBL25137217 0.64 PARP15 (0.44) MAPTNPC1SMN1; SMN2HTTPRNP
SCHEMBL16608505 0.64 CYP2A6 (0.36) KDM4ECYP2A6HTR3EHTR3BHTR3A
SCHEMBL10657900 0.63 PRNP (0.37) MAPTNPC1RAB9ASMN1; SMN2CYP2A6
SCHEMBL15643529 0.63 PSMB8 (0.52) MAPTKDM4ESMN1; SMN2HTTPOLB
SCHEMBL25322717 0.61 TNKS2 (0.57) MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4786633-A HIGHER ACTIVITY TANABE SEIYAKU CO., LTD. (JP) 1988-11-22 US disclosed
EP-0248645-A2 Cephalosporin compounds Tanabe Seiyaku Co., Ltd. (JP) 1987-12-09 EP disclosed