SCHEMBL10659380

SCHEMBL10659380

O=C(O)CC(Br)CCCBr

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
SLC22A6 Q4U2R8 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
GPR84 Q9NQS5 4/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
FOLH1 Q04609 1/20 0.33
GABRR1 P24046 2/20 0.31
LMNA P02545 1/20 0.31
LCK P06239 1/20 0.30
PPARD Q03181 1/20 0.30
ZDHHC20 Q5W0Z9 1/20 0.30
ZDHHC2 Q9UIJ5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474509 0.93 TSHR (0.39) TSHRSLC22A6TDP1GPR84ALDH1A1
SCHEMBL6829382 0.91 GPR84 (0.39) TSHRSLC22A6TDP1GPR84ALDH1A1
SCHEMBL4844058 0.81 LMNA (0.46) TSHRSLC22A6GPR84FOLH1GABRR1
SCHEMBL28099127 0.79 SLC22A6 (0.35) TSHRSLC22A6TDP1GPR84SMN1; SMN2
SCHEMBL6464981 0.79 GPR84 (0.50) TSHRSLC22A6TDP1GPR84ALDH1A1
SCHEMBL23829834 0.79 LMNA (0.43) TSHRSLC22A6GPR84FOLH1GABRR1
SCHEMBL6463034 0.77 GPR84 (0.59) TSHRSLC22A6TDP1GPR84ALDH1A1
SCHEMBL6460749 0.77 BLM (0.45) SLC22A6GPR84LMNALCKPPARD
SCHEMBL6465807 0.77 BLM (0.41) SLC22A6GPR84LMNALCKPPARD
SCHEMBL666360 0.76 GPR84 (0.57) TSHRSLC22A6TDP1GPR84SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210289794-A1 COMPOSITIONS AND RELATED METHODS FOR AGRICULTURE FLAGSHIP PIONEERING INNOVATIONS V, INC. 2021-09-23 US disclosed
EP-0090516-B1 SUBSTITUTED HEXAHYDROPYRROLO(1,2-A)-QUINOLINE, HEXAHYDRO-1H-PYRIDO(1,2-A)-QUINOLINE, HEXAHYDROBENZO(3)INDENE AND OCTAHYDROPHENANTHRENE CNS AGENTS PFIZER INC. (US) 1988-07-06 EP disclosed
US-4576964-A ANALGESICS, ANTIEMETICS PFIZER INC. (US) 1986-03-18 US disclosed
US-4476131-A ANTIEMETICS, ANALGESICS PFIZER INC. (US) 1984-10-09 US disclosed
EP-0090516-A1 Substituted hexahydropyrrolo(1,2-a)-quinoline, hexahydro-1H-pyrido(1,2-a)-quinoline, hexahydrobenzo(3)indene and octahydrophenanthrene CNS agents PFIZER INC. (US) 1983-10-05 EP disclosed