SCHEMBL10663333

SCHEMBL10663333

CC1=C(CC(=O)O)C(c2ccccc2Cl)C(C(=O)O)=C(C)N1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
HSD17B10 Q99714 4/20 0.43
TSHR P16473 3/20 0.43
HPGD P15428 3/20 0.43
MAPT P10636 2/20 0.43
CASP1 P29466 2/20 0.43
CASP7 P55210 2/20 0.43
ALOX15 P16050 1/20 0.43
POLB P06746 1/20 0.42
CYP2C9 P11712 3/20 0.41
KDM4E B2RXH2 3/20 0.41
TBXA2R P21731 3/20 0.41
ADRA1A P35348 3/20 0.41
SLC6A3 Q01959 3/20 0.41
MEN1 O00255 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
KMT2A Q03164 2/20 0.41
HIF1A Q16665 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL819493 0.90 CYP2C9 (0.53) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL7376559 0.90 CYP2C9 (0.53) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL7373610 0.90 CYP2C9 (0.53) ALDH1A1HSD17B10TSHRHPGDMAPT
Phenylpiperazine SCHEMBL10666908 0.86 HTR6 (0.41) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL3034308 0.86 ALDH1A1 (0.49) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL10733597 0.83 TSHR (0.39) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL10666914 0.79 TSHR (0.39) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL7267559 0.78 TSHR (0.44) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL7273568 0.78 CYP2C9 (0.67) ALDH1A1HSD17B10TSHRHPGDMAPT
SCHEMBL7265615 0.77 ALDH1A1 (0.43) ALDH1A1HSD17B10TSHRHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4753936-A CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1988-06-28 US disclosed
EP-0234196-A1 Substituted 1,4-dihydropyridine-3-carboxylic acid piperazides, process for their preparation and their use in medicaments BAYER AG (DE) 1987-09-02 EP disclosed