SCHEMBL10663545

SCHEMBL10663545

O=[N+]([O-])c1cccc(NCCNCC(O)c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.49
ADRB1 P08588 3/20 0.49
ADRB3 P13945 3/20 0.49
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DDX3X O00571 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10668067 0.91 ADRB2 (0.43) ADRB2ADRB1ADRB3ALDH1A1MEN1
SCHEMBL10667143 0.90 HIF1A (0.49) ADRB2ADRB1ADRB3ALDH1A1MEN1
SCHEMBL5605106 0.89 ALDH1A1 (0.53) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL11230234 0.81 ADRB1 (0.66) ADRB2ADRB1ADRB3ALDH1A1MEN1
Hydrochloric Acid SCHEMBL11247359 0.80 ADRB1 (0.68) ADRB2ADRB1ADRB3ALDH1A1MEN1
SCHEMBL10663547 0.77 ALDH1A1 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL11743087 0.77 MEN1 (0.52) ALDH1A1MEN1KMT2ASMN1; SMN2L3MBTL1
SCHEMBL11164763 0.76 ALDH1A1 (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL8975021 0.76 MAPT (0.57) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL18138767 0.75 MAPT (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4721717-A α-(aminoalkylaminomethyl)phenylmethanols, composition containing them, and use thereof to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-01-26 US disclosed
EP-0171689-B1 AMINOALCOHOLS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE COMPOUNDS AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1987-11-11 EP disclosed
EP-0171689-A1 Aminoalcohols, process for their preparation and medicaments containing these compounds and intermediates Roche Diagnostics GmbH (DE) 1986-02-19 EP disclosed