SCHEMBL10666131

SCHEMBL10666131

Cn1c2c(c3cc(F)ccc31)C(=O)CCC2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
KDM4E B2RXH2 2/20 0.43
PTGS1 P23219 4/20 0.43
PTGS2 P35354 4/20 0.43
ATM Q13315 1/20 0.41
MAPT P10636 1/20 0.40
ALOX5 P09917 1/20 0.39
MEN1 O00255 1/20 0.38
HCRTR1 O43613 1/20 0.38
KMT2A Q03164 1/20 0.38
SCARB1 Q8WTV0 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9596923 0.90 ATM (0.47) HDAC1HDAC6KDM4EPTGS1PTGS2
SCHEMBL10658421 0.84 KDM4E (0.43) HDAC1HDAC6KDM4EPTGS1PTGS2
SCHEMBL9596229 0.81 ALDH1A1 (0.50) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL10664163 0.81 KDM4E (0.41) HDAC1HDAC6KDM4EPTGS1PTGS2
SCHEMBL10664295 0.80 SCARB1 (0.42) KDM4EPTGS1PTGS2MAPTALOX5
SCHEMBL1146660 0.80 HTR2A (0.51) HDAC1HDAC6KDM4EALDH1A1
SCHEMBL30223533 0.80 HTR2A (0.51) HDAC1HDAC6KDM4EALDH1A1
SCHEMBL10667198 0.79 KDM4E (0.48) HDAC1HDAC6KDM4EPTGS1PTGS2
SCHEMBL7292545 0.78 PARP1 (0.45) ATM
SCHEMBL13877233 0.76 ALOX5 (0.65) PTGS1PTGS2ALOX5MEN1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4725615-A SELECTIVE FOR \"NEURONAL\" 5-HYDROXYTRYPTAMINE RECEPTORS; NERVOUS SYSTEM DISORDERS GLAXO GROUP LIMITED 1988-02-16 US disclosed
EP-0219193-A1 Tetrahydrocarbazolone derivatives, processes for their preparation and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1987-04-22 EP disclosed