SCHEMBL10666142

SCHEMBL10666142

CN(CCCN1CCc2cc3c(cc2C(=O)C1=O)OCO3)CCc1cc2ccccc2o1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 2/20 0.36
DRD5 P21918 1/20 0.36
CYP2D6 P10635 2/20 0.34
MAPT P10636 1/20 0.34
HCN4 Q9Y3Q4 1/20 0.34
DRD2 P14416 6/20 0.34
HTR2B P41595 5/20 0.34
CYP3A4 P08684 2/20 0.34
ALOX15 P16050 1/20 0.34
BCHE P06276 2/20 0.34
DRD3 P35462 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
GRM5 P41594 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624609 0.86 ADAM17 (0.34) DRD1DRD2HTR2BDRD3
SCHEMBL9624914 0.83 SIGMAR1 (0.34) DRD1DRD5CYP2D6MAPTHCN4
SCHEMBL9624838 0.81 HCN4 (0.51) MAPTHCN4DRD2HTR2BCYP3A4
Hydrochloric Acid SCHEMBL9624535 0.80 CYP3A4 (0.51) MAPTHCN4DRD2HTR2BCYP3A4
SCHEMBL9623990 0.77 SIGMAR1 (0.36) DRD1DRD5MAPTHCN4DRD2
SCHEMBL10667423 0.76 HCN4 (0.51) DRD1DRD5MAPTHCN4DRD2
SCHEMBL9623765 0.75 GNRHR (0.38) DRD1DRD5CYP2D6MAPTHCN4
SCHEMBL9624622 0.75 GNRHR (0.46) DRD1DRD5CYP2D6MAPTHCN4
SCHEMBL10667609 0.74 MAPT (0.42) MAPTHCN4CYP3A4ALOX15BCHE
SCHEMBL10668945 0.74 HCN4 (0.34) DRD1MAPTHCN4DRD2HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4737495-A ANTIALLERGENS, ANTISCHEMIC, HYPOTENSIVE AGENTS DR. KARL TOMAE, GMBH (DE) 1988-04-12 US disclosed
EP-0204349-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1986-12-10 EP disclosed