SCHEMBL10667759

SCHEMBL10667759

N#Cc1ccc(CCC(O)c2ccc(C#N)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.53
MMP13 P45452 2/20 0.53
CYP19A1 P11511 9/20 0.47
KCNJ1 P48048 1/20 0.44
KCNH2 Q12809 1/20 0.44
LOXL2 Q9Y4K0 2/20 0.44
CYP2A6 P11509 1/20 0.44
LSS P48449 1/20 0.44
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADRB2 P07550 1/20 0.41
DAO P14920 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109000 0.92 CYP19A1 (0.54) MMP12MMP13CYP19A1KCNH2LSS
SCHEMBL4084185 0.82 LOXL2 (0.48) MMP12MMP13CYP19A1KCNJ1KCNH2
SCHEMBL13891122 0.81 CA12 (0.41) MMP12MMP13CYP19A1LOXL2CYP2A6
SCHEMBL3656126 0.79 MMP12 (0.54) MMP12MMP13CYP19A1KCNJ1KCNH2
SCHEMBL11980400 0.79 CA12 (0.43) MMP12MMP13CYP19A1LOXL2CYP2A6
SCHEMBL9647636 0.78 TSHR (0.45) CYP19A1CYP2A6TSHRHSD17B10
SCHEMBL2964767 0.76 ADRB2 (0.62) TSHRADRB2
SCHEMBL13174142 0.76 CA12 (0.44) CYP19A1LOXL2CYP2A6TSHR
SCHEMBL11980418 0.76 CA12 (0.44) CYP19A1LOXL2CYP2A6TSHR
SCHEMBL28239877 0.76 CA12 (0.44) CYP19A1LOXL2CYP2A6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4732907-A Antiprotozoal diamidines and bis-imidazoline PFIZER INC. (US) 1988-03-22 US disclosed
US-4624958-A Antiprotozoal 1,4-di(p-amidinophenyl)imidazoles PFIZER INC. (US) 1986-11-25 US disclosed
US-4546113-A Antiprotozoal diamidines PFIZER INC. (US) 1985-10-08 US disclosed