SCHEMBL10668261

SCHEMBL10668261

N#Cc1ccc(CC(O)Cc2ccc(C#N)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.52
CYP2A6 P11509 2/20 0.52
MMP12 P39900 1/20 0.47
MMP13 P45452 1/20 0.47
CA12 O43570 1/20 0.46
CA2 P00918 1/20 0.46
CA3 P07451 1/20 0.46
CA6 P23280 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
IDO1 P14902 2/20 0.46
HRH3 Q9Y5N1 1/20 0.44
SAE1 Q9UBE0 1/20 0.43
UBA2 Q9UBT2 1/20 0.43
HTT P42858 1/20 0.43
CYP19A1 P11511 2/20 0.42
KCNJ1 P48048 1/20 0.42
KCNH2 Q12809 1/20 0.42
CTBP2 P56545 1/20 0.42
MMP3 P08254 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10621501 0.88 CYP2A6 (0.55) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL7395294 0.85 LOXL2 (0.42) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL1226223 0.84 LOXL2 (0.50) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL379566 0.83 CYP2A6 (0.54) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL19354446 0.83 CYP2A6 (0.54) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL4084185 0.83 LOXL2 (0.48) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL19143772 0.82 MMP12 (0.43) LOXL2CYP2A6MMP12MMP13HRH3
SCHEMBL19354445 0.79 CYP2A6 (0.50) LOXL2CYP2A6MMP12MMP13CA12
SCHEMBL92970 0.78 LOXL2 (0.58) LOXL2CYP2A6CA12CA2CA3
SCHEMBL6245764 0.78 KDM6B (0.51) LOXL2CYP2A6MMP12MMP13CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4732907-A Antiprotozoal diamidines and bis-imidazoline PFIZER INC. (US) 1988-03-22 US disclosed
US-4624958-A Antiprotozoal 1,4-di(p-amidinophenyl)imidazoles PFIZER INC. (US) 1986-11-25 US disclosed
US-4546113-A Antiprotozoal diamidines PFIZER INC. (US) 1985-10-08 US disclosed