SCHEMBL10669484

SCHEMBL10669484

CCOC(=O)Nc1ccc(N(F)Cc2ccccc2)nc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 5/20 0.50
KCNQ3 O43525 4/20 0.50
CYP1A2 P05177 3/20 0.50
CYP2C9 P11712 3/20 0.50
CYP2C19 P33261 3/20 0.50
HSD17B10 Q99714 3/20 0.50
NFKB1 P19838 2/20 0.50
ABCB11 O95342 1/20 0.50
ESR1 P03372 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CYP2D6 P10635 1/20 0.50
ALOX15 P16050 1/20 0.50
TBXA2R P21731 1/20 0.50
MAPK1 P28482 1/20 0.50
CASP1 P29466 1/20 0.50
SHMT2 P34897 1/20 0.50
PTGS2 P35354 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1826738 0.81 KCNQ2 (0.60) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL15004036 0.79 KCNQ2 (0.63) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL29754311 0.75 KCNQ3 (0.79) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL10791137 0.75 KCNQ3 (0.79) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL10790424 0.74 KCNQ3 (0.77) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL21623758 0.74 ALDH1A1 (0.50) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL20654769 0.74 CYP1A2 (0.62) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
SCHEMBL14638232 0.73 PKM (0.50) KCNQ2CYP1A2CYP2C9CYP2C19NFKB1
SCHEMBL19700168 0.71 KCNQ2 (0.45) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Maleic Acid SCHEMBL5381020 0.71 ALDH1A1 (0.63) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778799-A ANALGESIC, ANTIPYRETIC, ANTIINFLAMMATORY AGENT TIBES ULRICH (DE) 1988-10-18 US disclosed