SCHEMBL10669696

SCHEMBL10669696

Cc1nccn1-c1ccc(C(=O)CCC(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
PDE4A P27815 2/20 0.51
PDE4B Q07343 2/20 0.51
PDE4C Q08493 2/20 0.51
PDE4D Q08499 2/20 0.51
ALDH1A1 P00352 4/20 0.50
PDE3B Q13370 1/20 0.50
PDE3A Q14432 1/20 0.50
POLB P06746 1/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2D6 P10635 3/20 0.47
CYP1A2 P05177 3/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP19A1 P11511 1/20 0.47
NR4A2 P43354 2/20 0.46
NR4A1 P22736 1/20 0.46
USP5 P45974 1/20 0.45
PORCN Q9H237 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12589742 0.84 ALDH1A1 (0.50) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL17116879 0.84 PDE4A (0.56) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL8297463 0.82 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL10672237 0.82 SMN1; SMN2 (0.55) KMT2AALDH1A1POLBCYP3A4CYP2D6
SCHEMBL326869 0.82 NR4A1 (0.65) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL16198288 0.81 ALDH1A1 (0.51) PDE4APDE4BPDE4CPDE4DALDH1A1
Hydrochloric Acid SCHEMBL6947520 0.81 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL1839310 0.81 PDE4A (0.47) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL28186274 0.80 NR4A1 (0.63) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL30831804 0.80 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4734415-A CARDIOTONIC, HYPOTENSIVE WARNER-LAMBERT COMPANY (US) 1988-03-29 US disclosed
US-4353905-A CARDIOTONIC AGENTS WARNER-LAMBERT COMPANY (US) 1982-10-12 US disclosed