SCHEMBL10670569

SCHEMBL10670569

Brc1ccc2c(c1)c1ccccc1n2CC#CC#CCn1c2ccccc2c2cc(Br)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSPO P30536 3/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
RAD52 P43351 1/20 0.48
POLB P06746 1/20 0.44
MAPT P10636 4/20 0.44
TP53 P04637 1/20 0.43
DNM1 Q05193 5/20 0.43
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
HBB P68871 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8335552 0.84 CYP1A2 (0.56) MEN1KMT2APOLBMAPTALDH1A1
SCHEMBL11493115 0.84 TSPO (0.50) TSPOMEN1KMT2ARAD52POLB
SCHEMBL29773622 0.78 MAPT (0.65) TSPOMEN1KMT2ARAD52POLB
SCHEMBL871044 0.78 MAPT (0.65) TSPOMEN1KMT2ARAD52POLB
SCHEMBL29696470 0.77 MAOA (0.53) TSPOMEN1KMT2ARAD52
SCHEMBL2456180 0.76 POLB (0.53) TSPOMEN1KMT2APOLBMAPT
SCHEMBL10954372 0.75 TSPO (0.51) TSPOMEN1KMT2ARAD52MAPT
SCHEMBL17955864 0.75 MAPT (0.58) TSPOMEN1KMT2ARAD52POLB
SCHEMBL2246814 0.75 CYP19A1 (0.70) TSPOMEN1KMT2ARAD52MAPT
SCHEMBL1921157 0.75 ALDH1A1 (0.60) TSPOMEN1KMT2ARAD52POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4743659-A Chemical modification of polydiacetylene crystals GTE LABORATORIES INCORPORATED (US) 1988-05-10 US disclosed
US-4681920-A Chemical modification of polydiacetylene crystals GTE LABORATORIES INCORPORATED (US) 1987-07-21 US disclosed
US-4208501-A PHOTOCONDUCTORS AND OPTICAL DEVICES ALLIED CHEMICAL CORPORATION (US) 1980-06-17 US disclosed
US-4125534-A HIGH ENERGY RADIATION DOSAGE INDICATORS ALLIED CHEMICAL CORPORATION (US) 1978-11-14 US disclosed