SCHEMBL1067537

SCHEMBL1067537

CCC1CCc2c(sc(N)c2C(N)=O)C1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.80
MAPT P10636 13/20 0.80
HPGD P15428 10/20 0.72
GAA P10253 3/20 0.72
KDM4E B2RXH2 12/20 0.68
HSD17B10 Q99714 5/20 0.68
ALOX15 P16050 4/20 0.68
SMN1; SMN2 Q16637 4/20 0.64
LMNA P02545 2/20 0.64
ANO1 Q5XXA6 1/20 0.63
AIP O00170 1/20 0.62
SGTA O43765 1/20 0.62
TOMM70 O94826 1/20 0.62
STIP1 P31948 1/20 0.62
PPP5C P53041 1/20 0.62
DNAJC7 Q99615 1/20 0.62
STUB1 Q9UNE7 1/20 0.62
TNIK Q9UKE5 1/20 0.57
RAB9A P51151 2/20 0.54
MEN1 O00255 6/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17189283 0.89 ALDH1A1 (0.72) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL14478808 0.84 ALDH1A1 (1.00) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL1718839 0.81 MAPT (1.00) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL5451299 0.78 ALDH1A1 (0.60) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL5451294 0.78 ALDH1A1 (0.60) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL18220881 0.77 MAPT (0.68) ALDH1A1MAPTHPGDGAAKDM4E
SCHEMBL1719520 0.77 ALDH1A1 (1.00) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL5453282 0.76 AIP (0.71) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL5451446 0.76 AIP (0.71) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL5460515 0.76 AIP (0.69) ALDH1A1MAPTHPGDKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4683912-A1 SUBSTITUTED THIOPHENE FUSED CYCLOHEXANONE DERIVATIVES, COMPOSITIONS COMPRISING THE SAME AND THEIR USE AS PHARMACEUTICALS Neurasic Therapeutics Inc. (CA) 2026-01-28 EP disclosed
WO-2025035205-A1 PHARMACEUTICAL COMBINATIONS COMPRISING A SUBSTITUTED THIOPHENE FUSED CYCLOHEXANONE DERIVATIVE AND A CYCLOOXYGENASE (COX) INHIBITOR, AND THEIR USE FOR THE TREATMENT OF PAIN NEURASIC THERAPEUTICS INC. (CA) 2025-02-20 WO disclosed
WO-2024192520-A1 SUBSTITUTED THIOPHENE FUSED CYCLOHEXANONE DERIVATIVES, COMPOSITIONS COMPRISING THE SAME AND THEIR USE AS PHARMACEUTICALS NEURASIC THERAPEUTICS INC. (CA) 2024-09-26 WO disclosed
EP-2222326-B2 INHIBITORS OF MALT1 PROTEOLYTIC ACTIVITY AND USES THEREOF VIB VZW (BE) 2015-02-25 EP disclosed
EP-2222326-B1 Inhibitors of MALT1-proteolytic activity and uses thereof VIB VZW (BE) 2012-04-18 EP disclosed
US-20110021548-A1 INHIBITORS OF MALT1 PROTEOLYTIC ACTIVITY AND USES THEREOF UNIVERSITEIT GENT (BE) 2011-01-27 US disclosed
US-20110021548-A1 INHIBITORS OF MALT1 PROTEOLYTIC ACTIVITY AND USES THEREOF UNIVERSITEIT GENT (BE) 2011-01-27 US disclosed
US-20110021548-A1 INHIBITORS OF MALT1 PROTEOLYTIC ACTIVITY AND USES THEREOF UNIVERSITEIT GENT (BE) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021548-A1 INHIBITORS OF MALT1 PROTEOLYTIC ACTIVITY AND USES THEREOF MMEL1, CTRL, ZFR ALDH1A1 4353/4885MAPT 4436/4885HPGD 3987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.